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2-Aminothiazole derivatives as selective allosteric modulators of the protein kinase CK2.: Part 1: Identification of an allosteric binding site

CK2 is a ubiquitous Ser/Thr protein kinase involved in the control of various signaling pathways and is known to be constitutively active. In the present study, we identified aryl 2-aminothiazoles as a novel class of CK2 inhibitors, which displayed a non ATP-competitive mode of action and stabilized...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Bestgen, Benoît, Krimm, Isabelle, Kufareva, Irina, Kamal, Ahmed Ashraf Moustafa, Seetoh, Wei-Guang, Abell, Chris, Hartmann, Rolf W., Abagyan, Ruben, Cochet, Claude, Borgne, Marc Le, Engel, Matthias, Lomberget, Thierry
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7667462/
https://ncbi.nlm.nih.gov/pubmed/30689953
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.8b01766
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