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Crystal Structure and Inhibitor Identifications Reveal Targeting Opportunity for the Atypical MAPK Kinase ERK3

Extracellular signal-regulated kinase 3 (ERK3), known also as mitogen-activated protein kinase 6 (MAPK6), is an atypical member of MAPK kinase family, which has been poorly studied. Little is known regarding its function in biological processes, yet this atypical kinase has been suggested to play im...

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Библиографические подробности
Опубликовано в: :Int J Mol Sci
Главные авторы: Schröder, Martin, Filippakopoulos, Panagis, Schwalm, Martin P., Ferrer, Carla A., Drewry, David H., Knapp, Stefan, Chaikuad, Apirat
Формат: Artigo
Язык:Inglês
Опубликовано: MDPI 2020
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC7663056/
https://ncbi.nlm.nih.gov/pubmed/33114754
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21217953
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