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Discovery of histone deacetylase 3 (HDAC3)-specific PROTACs()

Histone deacetylases (HDACs) are validated drug targets for cancer treatment. Increased HDAC isozyme selectivity and novel strategies to inhibit HDAC activity could lead to safer and more effective drug candidates. Nonetheless, it is quite challenging to develop isozyme-specific HDACi due to the hig...

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Detalles Bibliográficos
Publicado en:Chem Commun (Camb)
Main Authors: Xiao, Yufeng, Wang, Jia, Zhao, Lisa Y., Chen, Xinyi, Zheng, Guangrong, Zhang, Xuan, Liao, Daiqing
Formato: Artigo
Idioma:Inglês
Publicado: 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7654701/
https://ncbi.nlm.nih.gov/pubmed/32840532
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0cc03243c
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