Carregant...

Discovery of histone deacetylase 3 (HDAC3)-specific PROTACs()

Histone deacetylases (HDACs) are validated drug targets for cancer treatment. Increased HDAC isozyme selectivity and novel strategies to inhibit HDAC activity could lead to safer and more effective drug candidates. Nonetheless, it is quite challenging to develop isozyme-specific HDACi due to the hig...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Chem Commun (Camb)
Autors principals: Xiao, Yufeng, Wang, Jia, Zhao, Lisa Y., Chen, Xinyi, Zheng, Guangrong, Zhang, Xuan, Liao, Daiqing
Format: Artigo
Idioma:Inglês
Publicat: 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7654701/
https://ncbi.nlm.nih.gov/pubmed/32840532
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0cc03243c
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!