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Structure-Based Inhibitor Discovery of Class I Histone Deacetylases (HDACs)

Class I histone deacetylases (HDACs) are promising targets for epigenetic therapies for a range of diseases such as cancers, inflammations, infections and neurological diseases. Although six HDAC inhibitors are now licensed for clinical treatments, they are all pan-inhibitors with little or no HDAC...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Luo, Yuxiang, Li, Huilin
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7700698/
https://ncbi.nlm.nih.gov/pubmed/33266366
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21228828
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