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Structure-Based Inhibitor Discovery of Class I Histone Deacetylases (HDACs)

Class I histone deacetylases (HDACs) are promising targets for epigenetic therapies for a range of diseases such as cancers, inflammations, infections and neurological diseases. Although six HDAC inhibitors are now licensed for clinical treatments, they are all pan-inhibitors with little or no HDAC...

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Dades bibliogràfiques
Publicat a:Int J Mol Sci
Autors principals: Luo, Yuxiang, Li, Huilin
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7700698/
https://ncbi.nlm.nih.gov/pubmed/33266366
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21228828
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