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TAMI-20. POLY(ADP-RIBOSE) GLYCOHYDROLASE INHIBITION SEQUESTERS NAD+ TO POTENTIATE THE METABOLIC LETHALITY OF ALKYLATING CHEMOTHERAPY IN IDH MUTANT TUMOR CELLS

Mutations in IDH1 or IDH2 characterize the majority of diffuse infiltrative gliomas of younger adulthood. DNA alkylator chemotherapy has proven to be an effective treatment for IDH mutant glioma, yet recurrences remain frequent and improved treatments are needed. Upon exposure of cancer cells to DNA...

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Bibliografske podrobnosti
izdano v:Neuro Oncol
Main Authors: Nagashima, Hiroaki, Lee, Christine, Tateishi, Kensuke, Higuchi, Fumi, Subramanian, Megha, Rafferty, Seamus, Melamed, Lisa, Miller, Julie, Wakimoto, Hiroaki, Cahill, Daniel
Format: Artigo
Jezik:Inglês
Izdano: Oxford University Press 2020
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7650933/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/noaa215.909
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