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Molecular determinants of ligand efficacy and potency in GPCR signaling

G protein-coupled receptors bind to extracellular ligands and drugs and modulate intracellular responses through conformational changes. Despite their importance as drug targets, the molecular origins of pharmacological properties such as efficacy (maximum signaling response) and potency (the ligand...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Science
Hauptverfasser: Heydenreich, Franziska M., Marti-Solano, Maria, Sandhu, Manbir, Kobilka, Brian K., Bouvier, Michel, Babu, M. Madan
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2023
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7615523/
https://ncbi.nlm.nih.gov/pubmed/38127743
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.adh1859
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