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Molecular determinants of ligand efficacy and potency in GPCR signaling

G protein-coupled receptors bind to extracellular ligands and drugs and modulate intracellular responses through conformational changes. Despite their importance as drug targets, the molecular origins of pharmacological properties such as efficacy (maximum signaling response) and potency (the ligand...

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Détails bibliographiques
Publié dans:Science
Auteurs principaux: Heydenreich, Franziska M., Marti-Solano, Maria, Sandhu, Manbir, Kobilka, Brian K., Bouvier, Michel, Babu, M. Madan
Format: Artigo
Langue:Inglês
Publié: 2023
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7615523/
https://ncbi.nlm.nih.gov/pubmed/38127743
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.adh1859
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