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Short peptide pharmacophores developed from protein phosphatase-1 disrupting peptides (PDPs)

PP1 is a major phosphoserine/threonine-specific phosphatase that is involved in diseases such as heart insufficiency and diabetes. PP1-disrupting peptides (PDPs) are selective modulators of PP1 activity that release its catalytic subunit, which then dephosphorylates nearby substrates. Recently, PDPs...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Fontanillo, Miriam, Trebacz, Malgorzata, Reinkemeier, Christopher D., Huerta, Daniela Avilés, Uhrig, Ulrike, Sehr, Peter, Köhn, Maja
Formato: Artigo
Idioma:Inglês
Publicado em: 2022
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7613447/
https://ncbi.nlm.nih.gov/pubmed/35525109
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2022.116785
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