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Functional Consequences of Pravastatin Isomerization on OATP1B1-Mediated Transport
Pravastatin acid (PVA) can be isomerized to its inactive metabolite 3′α-iso-pravastatin acid (3αPVA) under acidic pH conditions. Previous studies reported interindividual differences in circulating concentrations of PVA and 3αPVA. This study investigated the functional consequences of PVA isomerizat...
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| Publicat a: | Drug Metab Dispos |
|---|---|
| Autors principals: | , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
The American Society for Pharmacology and Experimental Therapeutics
2020
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7589943/ https://ncbi.nlm.nih.gov/pubmed/32892153 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.120.000122 |
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