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Functional Consequences of Pravastatin Isomerization on OATP1B1-Mediated Transport

Pravastatin acid (PVA) can be isomerized to its inactive metabolite 3′α-iso-pravastatin acid (3αPVA) under acidic pH conditions. Previous studies reported interindividual differences in circulating concentrations of PVA and 3αPVA. This study investigated the functional consequences of PVA isomerizat...

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Publicat a:Drug Metab Dispos
Autors principals: Wagner, Jonathan B., Ruggiero, Melissa, Leeder, J. Steven, Hagenbuch, Bruno
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7589943/
https://ncbi.nlm.nih.gov/pubmed/32892153
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.120.000122
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