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Synthesis and structure–activity relationship studies of novel dihydropyridones as androgen receptor modulators

A library of 3-hydroxy-2,3-dihyrdropyridones was synthesized and their activity as antiandrogens was tested in the human prostate cancer cell lines LNCaP. Structure–activity relationship studies resulted in the identification of a potent compound, whose activity is comparable to MDV3100. Homology mo...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Pepe, Antonella, Pamment, Michael, Kim, Yeong Sang, Lee, Sunmin, Lee, Min-Jung, Beebe, Kristin, Filikov, Anton, Neckers, Len, Trepel, Jane, Malhotra, Sanjay V.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7581280/
https://ncbi.nlm.nih.gov/pubmed/24044500
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301714s
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