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Inhibition, crystal structures, and in-solution oligomeric structure of aldehyde dehydrogenase 9A1

Aldehyde dehydrogenase 9A1 (ALDH9A1) is a human enzyme that catalyzes the NAD(+)-dependent oxidation of the carnitine precursor 4-trimethylaminobutyraldehyde to 4-N-trimethylaminobutyrate. Here we show that the broad-spectrum ALDH inhibitor diethylaminobenzaldehyde (DEAB) reversibly inhibits ALDH9A1...

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Publicat a:Arch Biochem Biophys
Autors principals: Wyatt, Jesse W., Korasick, David A., Qureshi, Insaf A., Campbell, Ashley C., Gates, Kent S., Tanner, John J.
Format: Artigo
Idioma:Inglês
Publicat: 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7484307/
https://ncbi.nlm.nih.gov/pubmed/32717224
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.abb.2020.108477
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