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Piperazine- and Piperidine-Containing Thiazolo[5,4-d]pyrimidine Derivatives as New Potent and Selective Adenosine A(2A) Receptor Inverse Agonists

The therapeutic use of A(2A) adenosine receptor (AR) antagonists for the treatment of neurodegenerative disorders, such as Parkinson and Alzheimer diseases, is a very promising approach. Moreover, the potential therapeutic role of A(2A) AR antagonists to avoid both immunoescaping of tumor cells and...

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Dettagli Bibliografici
Pubblicato in:Pharmaceuticals (Basel)
Autori principali: Varano, Flavia, Catarzi, Daniela, Vigiani, Erica, Vincenzi, Fabrizio, Pasquini, Silvia, Varani, Katia, Colotta, Vittoria
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7465344/
https://ncbi.nlm.nih.gov/pubmed/32722122
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph13080161
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