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Piperazine- and Piperidine-Containing Thiazolo[5,4-d]pyrimidine Derivatives as New Potent and Selective Adenosine A(2A) Receptor Inverse Agonists

The therapeutic use of A(2A) adenosine receptor (AR) antagonists for the treatment of neurodegenerative disorders, such as Parkinson and Alzheimer diseases, is a very promising approach. Moreover, the potential therapeutic role of A(2A) AR antagonists to avoid both immunoescaping of tumor cells and...

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Detalhes bibliográficos
Publicado no:Pharmaceuticals (Basel)
Main Authors: Varano, Flavia, Catarzi, Daniela, Vigiani, Erica, Vincenzi, Fabrizio, Pasquini, Silvia, Varani, Katia, Colotta, Vittoria
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7465344/
https://ncbi.nlm.nih.gov/pubmed/32722122
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph13080161
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