1,2,3-Triazolylmethaneboronate: A Structure Activity Relationship Study of a Class of β-Lactamase Inhibitors against Acinetobacter baumannii Cephalosporinase

[Image: see text] Boronic acid transition state inhibitors (BATSIs) are known reversible covalent inhibitors of serine β-lactamases. The selectivity and high potency of specific BATSIs bearing an amide side chain mimicking the β-lactam’s amide side chain are an established and recognized synthetic s...

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Vydáno v:ACS Infect Dis
Hlavní autoři: Caselli, Emilia, Fini, Francesco, Introvigne, Maria Luisa, Stucchi, Mattia, Taracila, Magdalena A., Fish, Erin R., Smolen, Kali A., Rather, Philip N., Powers, Rachel A., Wallar, Bradley J., Bonomo, Robert A., Prati, Fabio
Médium: Artigo
Jazyk:Inglês
Vydáno: American Chemical Society 2020
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7458062/
https://ncbi.nlm.nih.gov/pubmed/32502340
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.0c00254
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