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[(99m)Tc]Tc-DGA1, a Promising CCK(2)R-Antagonist-Based Tracer for Tumor Diagnosis with Single-Photon Emission Computed Tomography

Radiolabeled gastrin analogues have been proposed for theranostics of cholecystokinin subtype 2 receptor (CCK(2)R)-positive cancer. Peptide radioligands based on other receptor antagonists have displayed superior pharmacokinetics and higher biosafety than agonists. Here, we present DGA1, a derivativ...

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Detaylı Bibliyografya
Yayımlandı:Mol Pharm
Asıl Yazarlar: Kaloudi, Aikaterini, Kanellopoulos, Panagiotis, Radolf, Thorsten, Chepurny, Oleg G., Rouchota, Maritina, Loudos, George, Andreae, Fritz, Holz, George G., Nock, Berthold Artur, Maina, Theodosia
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7429258/
https://ncbi.nlm.nih.gov/pubmed/32568549
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.molpharmaceut.0c00605
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