Nalaganje...

Discovery of N-Substituted 2-Phenylcyclopropylmethylamines as Functionally Selective Serotonin 2C (5-HT(2C)) Receptor Agonists for Potential Use as Antipsychotic Medications

A series of N-substituted 2-phenylcyclopropylmethylamines were designed and synthesized, with the aim of finding 5-HT(2C)-selective agonists with preference for G(q) signaling. A number of these compounds exhibit 5-HT(2C) selectivity with preference for G(q)-mediated signaling compared with β-arrest...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
izdano v:J Med Chem
Main Authors: Zhang, Guiping, Cheng, Jianjun, McCorvy, John D., Lorello, Paul J., Caldarone, Barbara J., Roth, Bryan L., Kozikowski, Alan P.
Format: Artigo
Jezik:Inglês
Izdano: 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7374938/
https://ncbi.nlm.nih.gov/pubmed/28657744
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.7b00584
Oznake: Označite
Brez oznak, prvi označite!