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First‐in‐human study with ACT‐539313, a novel selective orexin‐1 receptor antagonist

AIMS: The orexin system is involved in anxiety behaviour and corresponding physiological reactions and constitutes a target for treatment of anxiety disorders. ACT‐539313 is a potent, selective orexin‐1 receptor antagonist being developed for the treatment of anxiety disorders. This first‐in‐human s...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Br J Clin Pharmacol
Egile Nagusiak: Kaufmann, Priska, Ort, Marion, Golor, Georg, Kornberger, Rüdiger, Dingemanse, Jasper
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: John Wiley and Sons Inc. 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7319015/
https://ncbi.nlm.nih.gov/pubmed/32067262
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.14251
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