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Increased Efficacy of Histone Methyltransferase G9a Inhibitors Against MYCN-Amplified Neuroblastoma

Targeted inhibition of proteins modulating epigenetic changes is an increasingly important priority in cancer therapeutics, and many small molecule inhibitors are currently being developed. In the case of neuroblastoma (NB), a pediatric solid tumor with a paucity of intragenic mutations, epigenetic...

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Détails bibliographiques
Publié dans:Front Oncol
Auteurs principaux: Bellamy, Jacob, Szemes, Marianna, Melegh, Zsombor, Dallosso, Anthony, Kollareddy, Madhu, Catchpoole, Daniel, Malik, Karim
Format: Artigo
Langue:Inglês
Publié: Frontiers Media S.A. 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7269128/
https://ncbi.nlm.nih.gov/pubmed/32537432
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2020.00818
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