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Increased Efficacy of Histone Methyltransferase G9a Inhibitors Against MYCN-Amplified Neuroblastoma

Targeted inhibition of proteins modulating epigenetic changes is an increasingly important priority in cancer therapeutics, and many small molecule inhibitors are currently being developed. In the case of neuroblastoma (NB), a pediatric solid tumor with a paucity of intragenic mutations, epigenetic...

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Detalhes bibliográficos
Publicado no:Front Oncol
Main Authors: Bellamy, Jacob, Szemes, Marianna, Melegh, Zsombor, Dallosso, Anthony, Kollareddy, Madhu, Catchpoole, Daniel, Malik, Karim
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7269128/
https://ncbi.nlm.nih.gov/pubmed/32537432
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2020.00818
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