New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII

[Image: see text] In the present study we investigated the structure–activity relationships of a new series of 4-[(3-ethyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides (EMAC10101a–m). All synthesized compounds, with the exception of compound EMAC10101k, preferentially inhibi...

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Publicat a:ACS Med Chem Lett
Autors principals: Meleddu, Rita, Distinto, Simona, Cottiglia, Filippo, Angius, Rossella, Caboni, Pierluigi, Angeli, Andrea, Melis, Claudia, Deplano, Serenella, Alcaro, Stefano, Ortuso, Francesco, Supuran, Claudiu T., Maccioni, Elias
Format: Artigo
Idioma:Inglês
Publicat: American Chemical Society 2020
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7236253/
https://ncbi.nlm.nih.gov/pubmed/32435395
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00644
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