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Active transport of rhodamine 123 by the human multidrug transporter P‐glycoprotein involves two independent outer gates

Human P‐glycoprotein (P‐gp) is a multispecific drug‐efflux transporter, which plays an important role in drug resistance and drug disposition. Recent cryo‐electron microscopy structures confirmed its rotationally symmetric architecture, which allows dual interaction with ATP and substrates. We here...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Pharmacol Res Perspect
Päätekijät: Nasim, Fauzia, Schmid, Diethart, Szakács, Gergely, Sohail, Azmat, Sitte, Harald H., Chiba, Peter, Stockner, Thomas
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: John Wiley and Sons Inc. 2020
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC7105846/
https://ncbi.nlm.nih.gov/pubmed/32232949
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.572
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