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Quantitative Proteomics of Clinically Relevant Drug-Metabolizing Enzymes and Drug Transporters and Their Intercorrelations in the Human Small Intestine

The levels of drug-metabolizing enzymes (DMEs) and transporter proteins in the human intestine are pertinent to determine oral drug bioavailability. Despite the paucity of reports on such measurements, it is well recognized that these values are essential for translating in vitro data on drug metabo...

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Dettagli Bibliografici
Pubblicato in:Drug Metab Dispos
Autori principali: Couto, Narciso, Al-Majdoub, Zubida M., Gibson, Stephanie, Davies, Pamela J., Achour, Brahim, Harwood, Matthew D., Carlson, Gordon, Barber, Jill, Rostami-Hodjegan, Amin, Warhurst, Geoffrey
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7076527/
https://ncbi.nlm.nih.gov/pubmed/31959703
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.119.089656
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