Nalaganje...

Organocatalytic Enantioselective Conjugate Addition of Nitromethane to Benzylidene-2-Benzoyl Acetate: Asymmetric Synthesis of ABT – 627, an Endothelin Receptor Antagonist

First catalytic and enantioselective conjugate addition of nitromethane to benzylidene-2-benzoyl acetate has been developed using dihydroquinine derived squaramide catalyst with moderate to high selectivities. Asymmetric total synthesis of ABT-627, a potent ETA receptor antagonist is accomplished ut...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
izdano v:Front Chem
Main Authors: Hajra, Saumen, Aziz, Sk Mohammad, Jana, Bibekananda, Hazra, Sunit
Format: Artigo
Jezik:Inglês
Izdano: Frontiers Media S.A. 2020
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7066299/
https://ncbi.nlm.nih.gov/pubmed/32195223
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2020.00135
Oznake: Označite
Brez oznak, prvi označite!