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Structure‐Based Design of a Macrocyclic PROTAC

Constraining a molecule in its bioactive conformation via macrocyclization represents an attractive strategy to rationally design functional chemical probes. While this approach has been applied to enzyme inhibitors or receptor antagonists, to date it remains unprecedented for bifunctional molecules...

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Detalhes bibliográficos
Publicado no:Angew Chem Int Ed Engl
Main Authors: Testa, Andrea, Hughes, Scott J., Lucas, Xavier, Wright, Jane E., Ciulli, Alessio
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7004083/
https://ncbi.nlm.nih.gov/pubmed/31746102
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201914396
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