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Allosteric Interactions in Human Cytochrome P450 CYP3A4: The Role of Phenylalanine 213

The role of Phe213 in the allosteric mechanism of human cytochrome P450 CYP3A4 was studied using a combination of progesterone (PGS) and carbamazepine (CBZ) as probe substrates. We expressed, purified and incorporated in POPC Nanodiscs three mutants, F213A, F213S, and F213Y, and compared them with t...

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Vydáno v:Biochemistry
Hlavní autoři: Denisov, Ilia G., Grinkova, Yelena V., Nandigrami, Prithviraj, Shekhar, Mrinal, Tajkhorshid, Emad, Sligar, Stephen G.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7003538/
https://ncbi.nlm.nih.gov/pubmed/30785734
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b01268
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