Wird geladen...

Allosteric Interactions in Human Cytochrome P450 CYP3A4: The Role of Phenylalanine 213

The role of Phe213 in the allosteric mechanism of human cytochrome P450 CYP3A4 was studied using a combination of progesterone (PGS) and carbamazepine (CBZ) as probe substrates. We expressed, purified and incorporated in POPC Nanodiscs three mutants, F213A, F213S, and F213Y, and compared them with t...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:Biochemistry
Hauptverfasser: Denisov, Ilia G., Grinkova, Yelena V., Nandigrami, Prithviraj, Shekhar, Mrinal, Tajkhorshid, Emad, Sligar, Stephen G.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2019
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7003538/
https://ncbi.nlm.nih.gov/pubmed/30785734
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b01268
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!