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Unleashing the full potential of Hsp90 inhibitors as cancer therapeutics through simultaneous inactivation of Hsp90, Grp94, and TRAP1

The Hsp90 family proteins Hsp90, Grp94, and TRAP1 are present in the cell cytoplasm, endoplasmic reticulum, and mitochondria, respectively; all play important roles in tumorigenesis by regulating protein homeostasis in response to stress. Thus, simultaneous inhibition of all Hsp90 paralogs is a reas...

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Publicado en:Exp Mol Med
Autores principales: Park, Hye-Kyung, Yoon, Nam Gu, Lee, Ji-Eun, Hu, Sung, Yoon, Sora, Kim, So Yeon, Hong, Jun-Hee, Nam, Dougu, Chae, Young Chan, Park, Jong Bae, Kang, Byoung Heon
Formato: Artigo
Lenguaje:Inglês
Publicado: Nature Publishing Group UK 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7000702/
https://ncbi.nlm.nih.gov/pubmed/31956271
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s12276-019-0360-x
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