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Trimethoprim: An Old Antibacterial Drug as a Template to Search for New Targets. Synthesis, Biological Activity and Molecular Modeling Study of Novel Trimethoprim Analogs

A new series of trimethoprim (TMP) analogs containing amide bonds (1–6) have been synthesized. Molecular docking, as well as dihydrofolate reductase (DHFR) inhibition assay were used to confirm their affinity to bind dihydrofolate reductase enzyme. Data from the ethidium displacement test showed the...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Wróbel, Agnieszka, Maliszewski, Dawid, Baradyn, Maciej, Drozdowska, Danuta
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6983048/
https://ncbi.nlm.nih.gov/pubmed/31892256
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25010116
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