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Bifunctional Small Molecule Ligands of K-Ras Induce Its Association with Immunophilin Proteins

Here we report the design, synthesis and characterization of bifunctional chemical ligands that induce the association of Ras with ubiquitously expressed immunophilin proteins such as FKBP12 and cyclophilin A. We show this approach is applicable to two distinct Ras ligand scaffolds, and that both th...

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Bibliografiset tiedot
Julkaisussa:Angew Chem Int Ed Engl
Päätekijät: Zhang, Ziyang, Shokat, Kevan M.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2019
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6980260/
https://ncbi.nlm.nih.gov/pubmed/31557383
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201910124
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