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Metabolism and Pharmacokinetic Study of the Boron-Containing Prodrug of Belinostat (ZL277), a Pan HDAC Inhibitor with Enhanced Bioavailability

ZL277 is a prodrug of belinostat with enhanced bioavailability and efficacy as a pan histone deacetylase (HDAC) inhibitor. In this study, we investigated the metabolism and pharmacokinetics of ZL277 in liver S9 fractions, liver microsomes, liver cytosol, and in mice. Metabolic products were identifi...

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Bibliografiske detaljer
Udgivet i:Pharmaceuticals (Basel)
Main Authors: Zhang, Changde, Guo, Shanchun, Zhong, Qiu, Zhang, Qiang, Hossain, Ahamed, Zheng, Shilong, Wang, Guangdi
Format: Artigo
Sprog:Inglês
Udgivet: MDPI 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6958523/
https://ncbi.nlm.nih.gov/pubmed/31817969
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph12040180
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