Загрузка...

Exploring Structural Determinants of Inhibitor Affinity and Selectivity in Complexes with Histone Deacetylase 6

Inhibition of histone deacetylase 6 (HDAC6) has emerged as a promising therapeutic strategy for the treatment of cancer, chemotherapy-induced peripheral neuropathy, and neurodegenerative disease. The recent X-ray crystal structure determination of HDAC6 enables an understanding of structural feature...

Полное описание

Сохранить в:
Библиографические подробности
Опубликовано в: :J Med Chem
Главные авторы: Osko, Jeremy D., Porter, Nicholas J., Reddy, Poli Adi Narayana, Xiao, You-Cai, Rokka, Johanna, Jung, Manfred, Hooker, Jacob M., Salvino, Joseph M., Christianson, David W.
Формат: Artigo
Язык:Inglês
Опубликовано: 2019
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6952581/
https://ncbi.nlm.nih.gov/pubmed/31793776
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b01540
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!