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Structural Determinants of Affinity and Selectivity in the Binding of Inhibitors to Histone Deacetylase 6

Histone deacetylase 6 (HDAC6) is associated with multiple neurological disorders as well as aggressive cancers, making its selective inhibition highly desirable for therapeutic purposes. The basic molecular design of an effective HDAC6 inhibitor consists of a zinc-binding group, a linker, and a capp...

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Bibliographic Details
Published in:Bioorg Med Chem Lett
Main Authors: Osko, Jeremy D., Christianson, David W.
Format: Artigo
Language:Inglês
Published: 2020
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7067655/
https://ncbi.nlm.nih.gov/pubmed/32067866
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2020.127023
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