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Methods for the expression, purification, and crystallization of histone deacetylase 6–inhibitor complexes

Histone deacetylase (HDAC) isozymes modulate numerous regulatory signals and pathways in biological systems, hence serving as targets for drug design. For example, HDAC6 is the cytosolic tubulin deacetylase and its inhibition compromises microtubule dynamics, leading to cancer cell cycle arrest and...

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Detaylı Bibliyografya
Yayımlandı:Methods Enzymol
Asıl Yazarlar: Osko, Jeremy D., Christianson, David W.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2019
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6941440/
https://ncbi.nlm.nih.gov/pubmed/31606087
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/bs.mie.2019.06.028
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