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Methods for the expression, purification, and crystallization of histone deacetylase 6–inhibitor complexes

Histone deacetylase (HDAC) isozymes modulate numerous regulatory signals and pathways in biological systems, hence serving as targets for drug design. For example, HDAC6 is the cytosolic tubulin deacetylase and its inhibition compromises microtubule dynamics, leading to cancer cell cycle arrest and...

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Dettagli Bibliografici
Pubblicato in:Methods Enzymol
Autori principali: Osko, Jeremy D., Christianson, David W.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6941440/
https://ncbi.nlm.nih.gov/pubmed/31606087
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/bs.mie.2019.06.028
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