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Targeted Protein Degradation: Elements of PROTAC Design

Targeted protein degradation using Proteolysis Targeting Chimeras (PROTACs) has emerged as a novel therapeutic modality in drug discovery. PROTACs mediate the degradation of select proteins of interest (POIs) by hijacking the activity of E3 ubiquitin ligases for POI ubiquitination and subsequent deg...

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Detalles Bibliográficos
Publicado en:Curr Opin Chem Biol
Main Authors: Paiva, Stacey-Lynn, Crews, Craig M.
Formato: Artigo
Idioma:Inglês
Publicado: 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6930012/
https://ncbi.nlm.nih.gov/pubmed/31004963
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cbpa.2019.02.022
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