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Fragment-based screening identifies molecules targeting the substrate-binding ankyrin repeat domains of tankyrase

The PARP enzyme and scaffolding protein tankyrase (TNKS, TNKS2) uses its ankyrin repeat clusters (ARCs) to bind a wide range of proteins and thereby controls diverse cellular functions. A number of these are implicated in cancer-relevant processes, including Wnt/β-catenin signalling, Hippo signallin...

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Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Pollock, Katie, Liu, Manjuan, Zaleska, Mariola, Meniconi, Mirco, Pfuhl, Mark, Collins, Ian, Guettler, Sebastian
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group UK 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6911004/
https://ncbi.nlm.nih.gov/pubmed/31836723
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-019-55240-5
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