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Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

The differential scanning fluorimetry (DSF) screening of 5.692 fragments in combination with benzenesulfonamide (BSA) against bovine carbonic anhydrase (bCA) delivered >100 hits that either caused, on their own, a significant thermal shift (ΔT(m), °C) in the protein melting temperature or signifi...

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Bibliografiset tiedot
Julkaisussa:J Enzyme Inhib Med Chem
Päätekijät: Krasavin, Mikhail, Kalinin, Stanislav, Zozulya, Sergey, Gryniukova, Anastasiia, Borysko, Petro, Angeli, Andrea, Supuran, Claudiu T.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Taylor & Francis 2019
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6896451/
https://ncbi.nlm.nih.gov/pubmed/31797704
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2019.1698562
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