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A systems pharmacokinetic/pharmacodynamic model for concizumab to explore the potential of anti-TFPI recycling antibodies

Concizumab is a humanized monoclonal antibody in clinical investigation directed against membrane-bound and soluble tissue factor pathway inhibitor (mTFPI and sTFPI) for treatment of hemophilia. Concizumab displays a non-linear pharmacokinetic (PK) profile due to mTFPI-mediated endocytosis and neces...

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Detalhes bibliográficos
Publicado no:Eur J Pharm Sci
Main Authors: Yuan, Dongfen, Rode, Frederik, Cao, Yanguang
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6824202/
https://ncbi.nlm.nih.gov/pubmed/31394258
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejps.2019.105032
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