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Design, Synthesis, and Biological Evaluation of Novel Thienopyrimidine Derivatives as PI3Kα Inhibitors

Three series of novel thienopyrimidine derivatives 9a–l, 15a–l, and 18a–h were designed and synthesized, and their IC(50) values against four cancer cell lines HepG-2, A549, PC-3, and MCF-7 were evaluated. Most compounds show moderate cytotoxicity against the tested cancer cell lines. The most promi...

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Vydáno v:Molecules
Hlavní autoři: Yu, Lide, Wang, Qinqin, Wang, Caolin, Zhang, Binliang, Yang, Zunhua, Fang, Yuanying, Zhu, Wufu, Zheng, Pengwu
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6804295/
https://ncbi.nlm.nih.gov/pubmed/31547116
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24193422
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