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Design, Synthesis, and Biological Evaluation of Novel Thienopyrimidine Derivatives as PI3Kα Inhibitors

Three series of novel thienopyrimidine derivatives 9a–l, 15a–l, and 18a–h were designed and synthesized, and their IC(50) values against four cancer cell lines HepG-2, A549, PC-3, and MCF-7 were evaluated. Most compounds show moderate cytotoxicity against the tested cancer cell lines. The most promi...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Yu, Lide, Wang, Qinqin, Wang, Caolin, Zhang, Binliang, Yang, Zunhua, Fang, Yuanying, Zhu, Wufu, Zheng, Pengwu
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6804295/
https://ncbi.nlm.nih.gov/pubmed/31547116
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24193422
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