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Structural Basis for the Regulation of PPARγ Activity by Imatinib

Imatinib is an effective anticancer drug for the treatment of leukemia. Interestingly, when an FDA-approved drug library was tested for agents that block peroxisome proliferator-activated receptor γ (PPARγ) phosphorylation at Ser245 to evaluate possibilities of antidiabetic drug repositioning, imati...

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Publicat a:Molecules
Autors principals: Jang, Jun Young, Kim, Hyun-Jung, Han, Byung Woo
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6803859/
https://ncbi.nlm.nih.gov/pubmed/31581474
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24193562
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