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Chlorpromazine Inhibits Miniature GABAergic Currents by Reducing the Binding and by Increasing the Unbinding Rate of GABA(A)Receptors

Recent studies have emphasized that nonequilibrium conditions of postsynaptic GABA(A) receptor (GABA(A)R) activation is a key factor in shaping the time course of IPSCs (Puia et al., 1994; Jones and Westbrook, 1995). Such nonequilibrium, resulting from extremely fast agonist time course, may affect...

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Pubblicato in:J Neurosci
Autori principali: Mozrzymas, Jerzy W., Barberis, Andrea, Michalak, Krystyna, Cherubini, Enrico
Natura: Artigo
Lingua:Inglês
Pubblicazione: Society for Neuroscience 1999
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6786064/
https://ncbi.nlm.nih.gov/pubmed/10087062
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.19-07-02474.1999
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