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Ortho-Methylarylamines as Time-Dependent Inhibitors of Cytochrome P450 1A1 Enzyme

Members of the cytochrome P450 1A family metabolize many procarcinogens such as polycyclic aromatic hydrocarbons and heterocyclic amines. Inactivation of these enzymes is a prerequisite for cancer prevention and treatment in certain cases. Mechanism-based inhibition (time and co-factor dependent) is...

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Detalhes bibliográficos
Publicado no:Drug Metab Lett
Main Authors: Sridhar, Jayalakshmi, Liu, Jiawang, Komati, Rajesh, Schroeder, Richard, Jiang, Quan, Tram, Phan, Riley, Kevin, Foroozesh, Maryam
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6697106/
https://ncbi.nlm.nih.gov/pubmed/28000546
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2174/1872312810666161220155226
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