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Targeting dynamic ATP-binding site features allows discrimination between highly homologous protein kinases

ATP-competitive inhibitors that demonstrate exquisite selectivity for specific members of the human kinome have been developed. Despite this success, the identification of highly selective inhibitors is still very challenging, and it is often not possible to rationally engineer selectivity between t...

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Pubblicato in:ACS Chem Biol
Autori principali: Chakraborty, Sujata, Inukai, Takayuki, Fang, Linglan, Golkowski, Martin, Maly, Dustin J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6642640/
https://ncbi.nlm.nih.gov/pubmed/31038916
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.9b00214
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