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Allosteric modulation of JNK docking-site interactions with ATP-competitive inhibitors

The c-Jun N-terminal kinases (JNKs) play a wide variety of roles in cellular signaling processes, dictating important, and even divergent, cellular fates. These essential kinases possess docking surfaces distal to their active sites that interact with diverse binding partners, including upstream act...

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Bibliografiske detaljer
Udgivet i:Biochemistry
Main Authors: Lombard, Chloe K., Davis, Audrey L., Inukai, Takayuki, Maly, Dustin J.
Format: Artigo
Sprog:Inglês
Udgivet: 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6338552/
https://ncbi.nlm.nih.gov/pubmed/30211540
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b00776
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