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Allosteric modulation of JNK docking-site interactions with ATP-competitive inhibitors

The c-Jun N-terminal kinases (JNKs) play a wide variety of roles in cellular signaling processes, dictating important, and even divergent, cellular fates. These essential kinases possess docking surfaces distal to their active sites that interact with diverse binding partners, including upstream act...

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Détails bibliographiques
Publié dans:Biochemistry
Auteurs principaux: Lombard, Chloe K., Davis, Audrey L., Inukai, Takayuki, Maly, Dustin J.
Format: Artigo
Langue:Inglês
Publié: 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6338552/
https://ncbi.nlm.nih.gov/pubmed/30211540
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b00776
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