A carregar...

Targeting dynamic ATP-binding site features allows discrimination between highly homologous protein kinases

ATP-competitive inhibitors that demonstrate exquisite selectivity for specific members of the human kinome have been developed. Despite this success, the identification of highly selective inhibitors is still very challenging, and it is often not possible to rationally engineer selectivity between t...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:ACS Chem Biol
Main Authors: Chakraborty, Sujata, Inukai, Takayuki, Fang, Linglan, Golkowski, Martin, Maly, Dustin J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6642640/
https://ncbi.nlm.nih.gov/pubmed/31038916
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.9b00214
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!