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What makes a kinase promiscuous for inhibitors?

ATP-competitive kinase inhibitors often bind several kinases due to the high conservation of the ATP binding pocket. Through clustering analysis of a large kinome profiling dataset we found a cluster of eight promiscuous kinases that on average bind more than five times more kinase inhibitors than t...

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Publicat a:Cell Chem Biol
Autors principals: Hanson, Sonya M., Georghiou, George, Thakur, Manish K., Miller, W. Todd, Rest, Joshua S., Chodera, John D., Seeliger, Markus A.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6632086/
https://ncbi.nlm.nih.gov/pubmed/30612951
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2018.11.005
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